Synthesis, characterization, inhibition effects, and molecular docking studies as acetylcholinesterase, α-glycosidase, and carbonic anhydrase inhibitors of novel benzenesulfonamides incorporating 1,3,5-triazine structural motifs | 2020/07/01 | English | 124 |
History of the development of antifungal azoles: A review on structures, SAR, and mechanism of action | 2020/11/01 | English | 124 |
Recent advancements of coumarin-based anticancer agents: An up-to-date review | 2020/10/01 | English | 122 |
Synthetic and medicinal perspective of thiazolidinones: A review | 2017/12/01 | English | 120 |
Design, synthesis and anticancer evaluation of thieno[2,3-d]pyrimidine derivatives as dual EGFR/HER2 inhibitors and apoptosis inducers | 2019/07/01 | English | 120 |
Novel antioxidant bromophenols with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions | 2017/10/01 | English | 119 |
Synthesis, molecular docking, acetylcholinesterase and butyrylcholinesterase inhibitory potential of thiazole analogs as new inhibitors for Alzheimer disease | 2015/10/01 | English | 117 |
The first synthesis of 4-phenylbutenone derivative bromophenols including natural products and their inhibition profiles for carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase enzymes | 2017/06/01 | English | 116 |
Novel 1,2,4-triazole derivatives as potential anticancer agents: Design, synthesis, molecular docking and mechanistic studies | 2018/02/01 | English | 115 |
Innovative nano-carriers in anticancer drug delivery-a comprehensive review | 2019/04/01 | English | 115 |
Investigation of inhibitory properties of some hydrazone compounds on hCA I, hCA II and AChE enzymes | 2019/05/01 | English | 114 |
Hydroxytyrosol lipophilic analogues: Enzymatic synthesis, radical scavenging activity and DNA oxidative damage protection | 2007/04/01 | English | 114 |
Design and synthesis of novel quinazolinone-1,2,3-triazole hybrids as new anti-diabetic agents: In vitro α-glucosidase inhibition, kinetic, and docking study | 2019/03/01 | English | 114 |
Novel thymol bearing oxypropanolamine derivatives as potent some metabolic enzyme inhibitors – Their antidiabetic, anticholinergic and antibacterial potentials | 2018/12/01 | English | 114 |
Quinolines, a perpetual, multipurpose scaffold in medicinal chemistry | 2021/04/01 | English | 111 |
Carbonic anhydrase inhibitory properties of novel benzylsulfamides using molecular modeling and experimental studies | 2014/10/01 | English | 111 |
Design, synthesis, molecular modeling, in vivo studies and anticancer evaluation of quinazolin-4(3H)-one derivatives as potential VEGFR-2 inhibitors and apoptosis inducers | 2020/01/01 | English | 111 |
Synthesis, characterization, crystal structure of novel bis-thiomethylcyclohexanone derivatives and their inhibitory properties against some metabolic enzymes | 2019/02/01 | English | 110 |
Synthesis, in vitro evaluation and molecular docking studies of thiazole derivatives as new inhibitors of α-glucosidase | 2015/10/01 | English | 110 |
Synthesis, biological evaluation and in silico studies of novel N-substituted phthalazine sulfonamide compounds as potent carbonic anhydrase and acetylcholinesterase inhibitors | 2019/08/01 | English | 109 |
The role of long noncoding RNA in major human disease | 2019/11/01 | English | 109 |
Promising anti-inflammatory effects of chalcones via inhibition of cyclooxygenase, prostaglandin E2, inducible NO synthase and nuclear factor κb activities | 2019/06/01 | English | 107 |
Design, synthesis, characterization, antimicrobial evaluation and molecular modeling studies of some dehydroacetic acid-chalcone-1,2,3-triazole hybrids | 2018/04/01 | English | 107 |
“Induced-fit”-type complex formation of the model enzyme α-cyclodextrin | 1976/06/01 | English | 105 |
Synthesis, molecular docking and anti-inflammatory screening of novel quinoline incorporated pyrazole derivatives using the Pfitzinger reaction II | 2015/02/01 | English | 105 |
Design, synthesis, molecular modeling and biological evaluation of novel 1H-pyrazolo[3,4-b]pyridine derivatives as potential anticancer agents | 2016/08/01 | English | 104 |
Estrogen receptor agonists/antagonists in breast cancer therapy: A critical review | 2017/04/01 | English | 104 |
The crystal and molecular structure of quercetin: A biologically active and naturally occurring flavonoid | 1986/03/01 | English | 104 |
Synthesis and bioactivities of pyrazoline benzensulfonamides as carbonic anhydrase and acetylcholinesterase inhibitors with low cytotoxicity | 2019/03/01 | English | 103 |
Encapsulation of ciprofloxacin within modified xanthan gum- chitosan based hydrogel for drug delivery | 2019/03/01 | English | 103 |