Current Drug Metabolism

Title Publication Date Language Citations
Neopterin as a Marker for Immune System Activation2002/04/01English492
The Cytochrome P450 Superfamily: Biochemistry, Evolution and Drug Metabolism in Humans2002/12/01English490
Drugs Behave as Substrates, Inhibitors and Inducers of Human Cytochrome P450 3A42008/05/01English452
A Comprehensive Listing of Bioactivation Pathways of Organic Functional Groups2005/06/01English415
Tyrosine Kinase Inhibitors – A Review on Pharmacology, Metabolism and Side Effects2009/06/01English411
UDP-Glucuronosyltransferases2000/09/01English371
(Section A: Molecular, Structural, and Cellular Biology of Drug Transporters) The MRP-Related and BCRP / ABCG2 Multidrug Resistance Proteins: Biology, Substrate Specificity and Regulation2004/02/01English346
Scaling Factors for the Extrapolation of In Vivo Metabolic Drug Clearance From In Vitro Data: Reaching a Consensus on Values of Human Micro-somal Protein and Hepatocellularity Per Gram of Liver2007/01/01English309
Medicinal Plants and Cancer Chemoprevention2008/09/01English296
Isothiocyanates as Cancer Chemopreventive Agents: Their Biological Activities and Metabolism in Rodents and Humans2002/06/01English295
Pharmacogenomics, Regulation and Signaling Pathways of Phase I and II Drug Metabolizing Enzymes2002/10/01English291
PEGylation of Proteins and Liposomes: a Powerful and Flexible Strategy to Improve the Drug Delivery2012/01/01English280
Incorporation of Pharmacogenomics into Routine Clinical Practice: the Clinical Pharmacogenetics Implementation Consortium (CPIC) Guideline Development Process2014/03/31English261
Prediction of Intestinal First-Pass Drug Metabolism2007/10/01English259
Design of Ester Prodrugs to Enhance Oral Absorption of Poorly Permeable Compounds: Challenges to the Discovery Scientist2003/12/01English238
Selective Serotonin Reuptake Inhibitors and Cytochrome P-450 Mediated Drug-Drug Interactions: An Update2002/02/01English235
A Microscale In Vitro Physiological Model of the Liver: Predictive Screens for Drug Metabolism and Enzyme Induction2005/12/01English228
The Metabolism and Toxicity of Quinones, Quinonimines, Quinone Methides, and Quinone-Thioethers2002/08/01English226
CYP2B6: New Insights into a Historically Overlooked Cytochrome P450 Isozyme2008/09/01English222
Xenobiotic-Induced Transcriptional Regulation of Xenobiotic Metabolizing Enzymes of the Cytochrome P450 Superfamily in Human Extrahepatic Tissues2008/02/01English215
Molecular Mechanisms Underlying the Dedifferentiation Process of Isolated Hepatocytes and Their Cultures2006/08/01English215
Cell Lines: A Tool for In Vitro Drug Metabolism Studies2008/01/01English211
Essential Oils: Extraction Techniques, Pharmaceutical And Therapeutic Potential - A Review2018/11/23English209
Cytochrome P450 Gene Polymorphism and Cancer2004/06/01English202
Metabolism of Green Tea Catechins: An Overview2006/10/01English202
The Conduct of Drug Metabolism Studies Considered Good Practice (II): In Vitro Experiments2007/12/01English200
L-Carnitine - Metabolic Functions and Meaning in Humans Life2011/09/01English197
Relevance of the Deletion Polymorphisms of the Glutathione S-Transferases GSTT1 and GSTM1 in Pharmacology and Toxicology2006/08/01English190
Evolutionary Advantage and Molecular Modes of Action of Multi-Component Mixtures Used in Phytomedicine2008/12/01English185
Structure and Function of the Human Breast Cancer Resistance Protein (BCRP/ABCG2)2010/09/01English184