Letters in Drug Design & Discovery

Title Publication Date Language Citations
Synthesis and Antifungal Activity of 1,3,4-Thiadiazole Derivatives Containing Pyridine Group2014/08/31English73
Synthesis, Antibacterial Activity of 2,4-Disubstituted Oxazoles and Thiazoles as Bioisosteres2009/01/01English73
Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities2017/04/06English71
Recent Developments in Natural and Synthetic Drug Research for Alzheimers Disease2006/05/01English61
New Heterocyclic Hydrazones in the Search for Antitubercular Agents: Synthesis and In Vitro Evaluations2006/09/01English54
Synthesis and Antifungal Activity of 1,2,3-thiadiazole Derivatives Containing 1,3,4-thiadiazole Moiety2014/06/01English53
Flexibility in the Molecular Design of Acetylcholinesterase Reactivators: Probing Representative Conformations by Chemometric Techniques and Docking/QM Calculations2016/04/14English51
Synthesis, Biological Evaluation and Docking Studies of 1,3,4-Oxadiazole Fused Benzothiazole Derivatives for Anticancer Drugs2018/12/01English51
Armed Imidazo [1,2-a] Pyrimidines (Pyridines): Evaluation of Antibacterial Activity2004/07/01English50
4-Hydroxy-3-methoxyphenyl Substituted 3-methyl-tetrahydroquinoline Derivatives Obtained Through Imino Diels-Alder Reactions as Potential Antitumoral Agents2010/11/01English48
Can Binding Kinetics Translate to a Clinically Differentiated Drug? From Theory to Practice2006/10/01English47
Synthesis and Biological Evaluation of Some Hydrazone Derivatives as Anti-inflammatory Agents2012/03/01English47
Szeged Index - Applications for Drug Modeling&#2005/12/01English42
Pt(II) vs Pd(II) Polyamine Complexes as New Anticancer Drugs: A Structure- Activity Study2006/04/01English41
Synthesis and Urease Inhibitory Properties of Some New N4-Substituted 5-Nitroisatin-3-thiosemicarbazones2010/02/01English40
Synthesis of Coumarin linked Naphthalimide Conjugates as Potential Anticancer and Antimicrobial Agents2009/04/01English39
In Vitro and In Vivo Investigations into the Carbene Silver Acetate Anticancer Drug Candidate SBC12012/09/01English39
Computationally Probing Drug-Protein Interactions Via Support Vector Machine2010/06/01English38
Physicochemical Interaction Study of Non-Steroidal Anti-Inflammatory Drugs with Dimyristoylphosphatidylethanolamine Liposomes2010/01/01English37
Recent Developments in the Synthesis and Applications of Anticancer Amonafide Derivatives. A Mini Review2015/10/30English37
Synthesis, Molecular Docking and Biological Evaluation of Mannich Products Based on Thiophene Nucleus using Ionic Liquid2018/11/29English35
In vitro Antimicrobial Activity of Liposomes Containing Ciprofloxacin,Meropenem and Gentamicin Against Gram-Negative Clinical Bacterial Strains2007/06/01English35
Synthesis and Antifungal Activity of 1,2,4-triazole Derivatives Containing Cyclopropane Moiety2012/04/26English34
Synthesis of 18F-labeled Neurotensin(8-13) via Copper-Mediated 1,3-Dipolar [3+2]Cycloaddition Reaction2007/06/01English33
Effect of the Metal Center on the Antitumor Activity of the Analogous Dinuclear Spermine Chelates (PdCl2)2(Spermine) and (PtCl2)2(Spermine)2007/10/01English33
Grid-Based Hydrogen Bond Potentials with Improved Directionality2004/04/01English33
Novel 1,3,4-Oxadiazole Fused Thiadiazole Derivatives: Synthesis and study of Anticancer Activities2019/05/24English32
Aminoalkylated Phenolic Chalcones: Investigation of Biological Effects on Acetylcholinesterase and Carbonic Anhydrase I and II as Potential Lead Enzyme Inhibitors2020/10/12English32
In Vitro and In Vivo Investigations into the Carbene Gold Chloride and Thioglucoside Anticancer Drug Candidates NHC-AuCl and NHC-AuSR2016/12/21English32
DPPH Scavenging Assay of Novel 1,3-disubstituted-1H-pyrazol-5-ols and their in silico Studies on Some Proteins Involved in Alzheimers Disease Signaling Cascade2010/03/01English31