Title	Publication Date	Language	Citations
The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints	2003/06/01	English	1,845
SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-β Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7	2002/07/01	English	1,268
Hypoxia-Inducible Factor-1 (HIF-1)	2006/08/03	English	1,138
G Protein-Coupled Receptors as Targets for Approved Drugs: How Many Targets and How Many Drugs?	2018/01/03	English	690
The Nuclear Receptor Peroxisome Proliferator-Activated Receptor-α Mediates the Anti-Inflammatory Actions of Palmitoylethanolamide	2004/10/01	English	660
Cloning and Functional Expression of the Human Histamine H3Receptor	1999/06/01	English	528
Differential Response of Estrogen Receptor α and Estrogen Receptor β to Partial Estrogen Agonists/Antagonists	1998/07/01	English	509
Neuroprotection against Oxidative Stress by Estrogens: Structure-Activity Relationship	1997/04/01	English	500
Nuclear Pregnane X Receptor and Constitutive Androstane Receptor Regulate Overlapping but Distinct Sets of Genes Involved in Xenobiotic Detoxification	2002/09/01	English	492
The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation ofCYP3A4by Rifampicin through a Distal Enhancer Module	1999/12/01	English	490
Inhibition of Transforming Growth Factor (TGF)-β1–Induced Extracellular Matrix with a Novel Inhibitor of the TGF-β Type I Receptor Kinase Activity: SB-431542	2002/07/01	English	480
Sex Differences in the Expression of Hepatic Drug Metabolizing Enzymes	2009/05/29	English	480
Altered Brain Serotonin Homeostasis and Locomotor Insensitivity to 3,4-Methylenedioxymethamphetamine (“Ecstasy”) in Serotonin Transporter-Deficient Mice	1998/04/01	English	472
dl-threo-β-Benzyloxyaspartate, A Potent Blocker of Excitatory Amino Acid Transporters	1998/02/01	English	449
The Cannabinoid CB1Receptor Antagonist SR141716 Increases Acrp30 mRNA Expression in Adipose Tissue of Obese fa/fa Rats and in Cultured Adipocyte Cells	2003/04/01	English	446
Amphetamine, 3,4-Methylenedioxymethamphetamine, Lysergic Acid Diethylamide, and Metabolites of the Catecholamine Neurotransmitters Are Agonists of a Rat Trace Amine Receptor	2001/12/01	English	440
Mechanisms of Release of Nucleotides and Integration of Their Action as P2X- and P2Y-Receptor Activating Molecules	2003/09/18	English	421
TAK-242 (Resatorvid), a Small-Molecule Inhibitor of Toll-Like Receptor (TLR) 4 Signaling, Binds Selectively to TLR4 and Interferes with Interactions between TLR4 and Its Adaptor Molecules	2010/09/29	English	400
Is Cisplatin-Induced Cell Death Always Produced by Apoptosis?	2001/04/01	English	397
Varenicline Is a Partial Agonist at α4β2 and a Full Agonist at α7 Neuronal Nicotinic Receptors	2006/06/09	English	391
(−)-Epigallocatechin-3-gallate Blocks the Induction of Nitric Oxide Synthase by Down-Regulating Lipopolysaccharide-Induced Activity of Transcription Factor Nuclear Factor-κB	1997/09/01	English	388
Curcumin (Diferuloylmethane) Down-Regulates Expression of Cell Proliferation and Antiapoptotic and Metastatic Gene Products through Suppression of IκBα Kinase and Akt Activation	2005/10/11	English	385
Evidence That Curcumin Suppresses the Growth of Malignant Gliomas in Vitro and in Vivo through Induction of Autophagy: Role of Akt and Extracellular Signal-Regulated Kinase Signaling Pathways	2007/03/29	English	379
The Repertoire of G-Protein–Coupled Receptors in Fully Sequenced Genomes	2005/02/01	English	374
Effector Pathway-Dependent Relative Efficacy at Serotonin Type 2A and 2C Receptors: Evidence for Agonist-Directed Trafficking of Receptor Stimulus	1998/07/01	English	363
Evidence for a New G Protein-Coupled Cannabinoid Receptor in Mouse Brain	2001/07/01	English	358
Multiple Amylin Receptors Arise from Receptor Activity-Modifying Protein Interaction with the Calcitonin Receptor Gene Product	1999/07/01	English	353
Identification and Characterization of Human Organic Anion Transporter 3 Expressing Predominantly in the Kidney	2001/05/01	English	353
NAD(P)H:Quinone Oxidoreductase 1: Role as a Superoxide Scavenger	2004/04/20	English	352
Characterization of SIS3, a Novel Specific Inhibitor of Smad3, and Its Effect on Transforming Growth Factor-β1-Induced Extracellular Matrix Expression	2005/11/15	English	341