Antileishmanial Activity of the Antiulcer Agent Omeprazole

Article Properties
  • Language
    English
  • Publication Date
    2002/08/01
  • Indian UGC (Journal)
  • Refrences
    19
  • Suping Jiang Department of Biological Sciences, University of Cincinnati, Cincinnati, Ohio 45221-0006
  • Juliana Meadows Department of Biological Sciences, University of Cincinnati, Cincinnati, Ohio 45221-0006
  • Steven A. Anderson Department of Biological Sciences, University of Cincinnati, Cincinnati, Ohio 45221-0006
  • Antony J. Mukkada Department of Biological Sciences, University of Cincinnati, Cincinnati, Ohio 45221-0006
Abstract
Cite
Jiang, Suping, et al. “Antileishmanial Activity of the Antiulcer Agent Omeprazole”. Antimicrobial Agents and Chemotherapy, vol. 46, no. 8, 2002, pp. 2569-74, https://doi.org/10.1128/aac.46.8.2569-2574.2002.
Jiang, S., Meadows, J., Anderson, S. A., & Mukkada, A. J. (2002). Antileishmanial Activity of the Antiulcer Agent Omeprazole. Antimicrobial Agents and Chemotherapy, 46(8), 2569-2574. https://doi.org/10.1128/aac.46.8.2569-2574.2002
Jiang S, Meadows J, Anderson SA, Mukkada AJ. Antileishmanial Activity of the Antiulcer Agent Omeprazole. Antimicrobial Agents and Chemotherapy. 2002;46(8):2569-74.
Journal Categories
Medicine
Public aspects of medicine
Toxicology
Poisons
Medicine
Therapeutics
Pharmacology
Science
Microbiology
Description

Could a common ulcer medication fight parasitic diseases? This research explores the antileishmanial activity of omeprazole, a widely used antiulcer drug, against *Leishmania donovani*, the causative agent of visceral leishmaniasis. The study reveals that omeprazole effectively inhibits the growth of promastigotes and amastigotes, demonstrating its potential as a novel therapeutic agent. Omeprazole's antiparasitic action stems from its inhibition of the P-type K+,H+-ATPase on the surface membrane of *Leishmania*. The drug is effective only at acidic pH, mimicking the conditions within phagolysosomal vesicles where the amastigote form resides. Promastigotes and amastigotes are reduced 90% or more with 150 μM omeprazole. These findings suggest that omeprazole may offer a less toxic alternative to existing chemotherapeutics for leishmaniasis. Its effectiveness at acidic pH makes it particularly promising, targeting the parasite within its natural environment. Further investigation is warranted to explore the clinical potential of omeprazole in treating visceral leishmaniasis.

Published in Antimicrobial Agents and Chemotherapy, this research aligns with the journal's focus on investigating and developing new antimicrobial agents. By demonstrating the antileishmanial activity of omeprazole, the study contributes to the journal's broader exploration of novel therapeutic strategies for infectious diseases. The citations reflect the paper's engagement with existing research in the fields of microbiology and pharmacology.

Refrences